Report error Found 172 of ki data for polymerid = 4500
Affinity DataKi: 0.180nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of human CHK1 expressed in baculovirus/insect cell systemMore data for this Ligand-Target Pair
Affinity DataKi: 1.75nM ΔG°: -11.8kcal/molepH: 7.4 T: 22°CAssay Description:The inhibitors reported in this study bind to CHK1 according to a general mechanism illustrated in Scheme 1 where E, S, and I stand for enzyme, subst...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 5.14nM ΔG°: -11.1kcal/molepH: 8.0 T: 20°CAssay Description:Surface plasmon resonance (SPR) biosensor binding studies were conducted using a Biacore 3000 instrument (GE Healtchare).More data for this Ligand-Target Pair
Affinity DataKi: 5.60nM ΔG°: -11.7kcal/molepH: 7.4 T: 37°CAssay Description:In vitro Chk1 enzymatic assay using purified enzyme, was incubated with substrate, and test compounds in the presence of 10 uM ATP/ [gamma-32P] ATP. ...More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:ChemBL affinity - Published Abbott papersMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Candidates for inhibitor selectivity characterization were chosen based on an initial single-timepoint commercial kinome profiling screen performed w...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of full length recombinant human N-terminal His-tagged CHK1 expressed in baculovirus infected Sf9 insect cells using CHK peptide as substr...More data for this Ligand-Target Pair